平安! 发表于 2011-11-9 19:57 9 u( T' D; k& _) b; ]" w0 E( Q. @
Pazopanib (100 mg/kg/day free base equivalent) % _6 S1 \4 M/ Z
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。3 X# ~3 \( I7 \, `% H4 ~
搜索了一下,原料一大堆。. e( p; u* X9 n" ]: w2 ^8 M
% h0 p2 @- c: U0 d( m) p对不起!100mg/kg是用于移植瘤的,我弄错了。
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1 H1 u c% n F+ r3 U以下是正版说明书的推荐用量。, ?3 Q5 A T7 a0 U1 S. z7 E
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--------------------- DOSAGE AND ADMINISTRATION ----------------
* A5 b' A6 m. w5 H5 i$ `- E* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
1 z# _, q; x) ~" Z* w, @* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) % h+ H% M! y( \
---------------------DOSAGE FORMS AND STRENGTHS --------------; M9 R. J) u/ b1 H; w
200 mg tablets. (3) 3 N/ g9 e, G5 x1 d1 g$ x
-------------------------------CONTRAINDICATIONS------------------------ |