平安! 发表于 2011-11-9 19:57 2 p1 V/ M* a q
Pazopanib (100 mg/kg/day free base equivalent) / q, G. I% x# j7 Q- T! \6 H
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。, s6 @- ?7 ?% J: p4 L1 w
搜索了一下,原料一大堆。( S! r: c% e) _1 Y+ q( a$ s
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对不起!100mg/kg是用于移植瘤的,我弄错了。7 m6 d& Y; y/ t3 k+ ~
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以下是正版说明书的推荐用量。8 \( E) L: ]: [- Z
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--------------------- DOSAGE AND ADMINISTRATION ----------------4 ]& [; {0 b& D# b& p0 ^) }
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) 0 n$ V' E) |( J7 |+ W
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
2 q5 Y* T4 j. E% @0 {, M1 n---------------------DOSAGE FORMS AND STRENGTHS --------------* Q& t8 D6 _* c
200 mg tablets. (3) * T$ S4 H& X- v- ^, N F
-------------------------------CONTRAINDICATIONS------------------------ |